KN-93 Phosphate 产品说明书 Chemicals
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产品编号 DC7180
名称 KN-93 Phosphate

化学性质

CAS 1188890-41-6
分子式 C26H29CLN2O4S.H3O4P
分子量 599.03
存储条件 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

生物活性

Description
In Vivo
In Vitro

化合物的使用

Kinase Assay
Cell Assay
Animal Administration

参考文献


KN-93 is a selective Ca2+/calmodulin-dependent protein kinase II inhibitor, which has been implicated in the regulation of smooth muscle contractility. CaM kinase II activation was inhibited by KN-93 pretreatment (IC50 ~1 μM). KN-93 inhibited histamine-in
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