VS-5584 产品说明书 Chemicals
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产品编号 DC7337
名称 VS-5584

化学性质

CAS 1246560-33-7
分子式 C17H22N8O
分子量 354.41
存储条件 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

生物活性

Description
In Vivo
In Vitro

化合物的使用

Kinase Assay
Cell Assay
Animal Administration

参考文献


VS-5584 is an ATP-competitive inhibitor which selectively inhibits PI3K/mTOR signaling with equivalent low nanomolar potency against all human Class I PI3K iso Forms and mTOR kinase. VS-5584 is approximately 10-fold selective For cancer stem cells with a
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