PP2(AGL 1879) 产品说明书 Chemicals
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产品编号 DC5008
名称 PP2(AGL 1879)

化学性质

CAS 172889-27-9
分子式 C15H16CLN5
分子量 301.77
存储条件 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

生物活性

Description
In Vivo
In Vitro

化合物的使用

Kinase Assay
Cell Assay
Animal Administration

参考文献


PP2 is a substance that has frequently been used in cancer research as a selective inhibitor For Src-family kinases. It strongly inhibits the kinases Lck (IC50=4 nM), Fyn (5 nM) and Hck (5 nM), shows weaker inhibition of EGFR (480 nM) and practically no
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