Dorsomorphin(BML-275) 产品说明书 Chemicals
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产品编号 DC8296
名称 Dorsomorphin(BML-275)

化学性质

CAS 866405-64-3
分子式 C24H25N5O
分子量 399.49
存储条件 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

生物活性

Description
In Vivo
In Vitro

化合物的使用

Kinase Assay
Cell Assay
Animal Administration

参考文献


Dorsomorphin(Compound C; BML-275) has been shown to act as a potent and selective inhibitor of AMPK (AMP-activated protein kinase; Ki = 109 nM), induced by AICAR and metformin; also inhibits the bone morphogenetic protein type 1 receptors ACTR-I (ALK2), B
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