BKM120 (NVP-BKM120, Buparlisib) 产品说明书 Chemicals
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产品编号 DC5154
名称 BKM120 (NVP-BKM120, Buparlisib)

化学性质

CAS 944396-07-0
分子式 C18H21F3N6O2
分子量 410.39
存储条件 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

生物活性

Description
In Vivo
In Vitro

化合物的使用

Kinase Assay
Cell Assay
Animal Administration

参考文献


Buparlisib, also known as BKM120, is an orally bioavailable specific oral inhibitor of the pan-class I phosphatidylinositol 3-kinase (PI3K) family of lipid kinases with potential antineoplastic activity. PI3K inhibitor BKM120 specifically inhibits class
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