Obicetrapib (AMG-899,TA-8995) 产品说明书 Chemicals
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产品编号 DC10134
名称 Obicetrapib (AMG-899,TA-8995)

化学性质

CAS 866399-87-3
分子式 C32H31F9N4O5
分子量 722.6
存储条件 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

生物活性

Description
In Vivo
In Vitro

化合物的使用

Kinase Assay
Cell Assay
Animal Administration

参考文献


Obicetrapib (also known as AMG-899, TA-8995, and DEX-001) is a cholesteryl ester transfer protein (CETP) inhibitor. CETP inhibitors substantially increase the concentration of high-density lipoprotein cholesterol (HDL-C), which may have a possible beneficial effect for cardiovascular disease risk reduction.
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