P22077

产品编号: DC7221 Featured
P22077
结构式
1247819-59-5
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中国地区超过5000个高品质化合物库存
应用领域
P 22077 是一种泛素蛋白特异性蛋白酶 (USP7) 抑制剂,EC50 值为 8.01 μM,同时可抑制 USP47,EC50 值为 8.74 μM。
Cas No.: 1247819-59-5
名称:
别名: P 22077; P-22077
SMILES: CC(=O)C1=CC(=C(S1)SC2=C(C=C(C=C2)F)F)[N+](=O)[O-]
分子式: C12H7F2NO3S2
分子量: 315.32
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: P22077 is an analog of the recently discovered USP7 inhibitor P5091. P22077 has negligible activity versus DEN1 and SENP2core over the concentration range tested, but inhibits USP7 with an IC50 of 8 μM. The inhibitory activities of P22077 in vitro agains
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
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MSDS_1627_DC7221_1247819-59-5
COA
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