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产品编号 产品名称 CAS No.
DC10114 Nifenalol

Nifenalol hydrochloride

5704-60-9
DC10115 Piperoxan hydrochloride

Piperoxan hydrochloride 是一种 α2 肾上腺素受体拮抗剂。

135-87-5
DC10384 Olodaterol

Olodaterol (BI1744)是长效的β2-adrenoceptor激动剂, EC50 值为1.4±0.08 nM。

868049-49-4
DC10683 DL 071-IT hydrochloride

7-[3-(tert-butylamino)-2-hydroxypropoxy]-3H-2-benzofuran-1-one,hydrochloride

55104-39-7
DC10693 O-Butyryl timolol

Butyryltimolol is a lipophilic ester prodrug of timolol, a beta adrenergic blocer with antihypertensive and hemodynamic properties.

106351-79-5
DC3172 Mirabegron

Mirabegron 是一种选择性的肾上腺素受体 (β3-adrenoceptor) 激动剂,EC50 为 22.4 nM。

223673-61-8
DC4240 Dexmedetomidine hydrochloride

Dexmedetomidine Hydrochloride 是α2肾上腺素受体激动剂,有止痛镇静活性。

145108-58-3
DC8436 Salmeterol Xinafoate

Salmeterol xinafoate 是长效 β2 肾上腺素能受体 (β2AR) 激动剂,对WT β2AR的Ki值为 1.5 nM。

94749-08-3
DC8583 Asenapine Maleate

Asenapine maleate是 5-HT(1A, 1B, 2A, 2B, 2C, 5A, 6, 7) 和 D2 的拮抗剂,Ki 值分别为 0.03-4.0 nM, 1.3 nM。同时也是一种抗精神病药物。

85650-56-2
DC8610 Salmeterol

Salmeterol是长效β2肾上腺素受体激动剂,可作用于哮喘。

89365-50-4
DC9248 Olodaterol(BI-1744) hydrochloride

Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptors located primarily in the lungs.

869477-96-3
DC9819 Guanoclor

Guanoclor is a sympatholytic drug. It is known to bind to non-adrenergic sites in pig kidney membranes.

5001-32-1
DC9333 Formoterol (Fumarate)

Formoterol fumarate(Foradil) is a potent, selective and long-acting β2-adrenoceptor agonist.

43229-80-7
DC8925 Atipamezole

Atipamezole(MPV1248) is an alpha-adrenoceptor antagonist with high affinity and selectivity for the alpha 2-receptor.

104054-27-5
DCAPI1411 Bisoprolol Fumarate

(±)-Bisoprolol hemifumarate is a selective β1-AR adrenergic antagonist. Possesses β1/β2 selectivity of approximately 100-fold and a Kd of 2-3 nM at the β1-AR (β1 receptor).

104344-23-2
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