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Cyclo(L-Pro-L-Val)

产品编号: DC26050 Featured
Cyclo(L-Pro-L-Val)
结构式
2854-40-2
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中国地区超过5000个高品质化合物库存
应用领域
Cyclo(L-Pro-L-Val) is a diketopiperazine that has been found in the marine sponge T. ignis, the bacterium B. pumilus, and the fungus A. fumigatus, among others.
化学性质生物活性化合物的使用COA & MSDS相关产品产品说明书
Cas No.: 2854-40-2
名称:
别名: Cyclo(L-prolyl-L-valine)
SMILES: O=C([C@H](C(C)C)N1)N2[C@](CCC2)([H])C1=O
分子式: C10H16N2O2
分子量: 196.2
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: Cyclo(L-Pro-L-Val) is a diketopiperazine that has been found in the marine sponge T. ignis, the bacterium B. pumilus, and the fungus A. fumigatus, among others.It is active against the bacteria S. aureus and B. subtilis (MICs = 16.3 and 18.2 µg/ml, respectively) but not E. coli (MIC = >20 µg/ml).Cyclo(L-Pro-L-Val) inhibits activation of a LuxR-dependent E. coli biosensor by the quorum-sensing molecule 3-oxo-hexanoyl-homoserine lactone (IC50 = 0.4 mM) and activates violacein pigment production in the LuxR-dependent C. violaceum acyl homoserine lactone reporter strain CV026.However, it does not activate or inhibit lacZ-based reporter fusions in S. liquefaciens or A. tumefaciens.
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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