TCS JNK 5a(JNK Inhibitor IX)

产品编号: DC8093 Featured
TCS JNK 5a(JNK Inhibitor IX)
结构式
312917-14-9
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中国地区超过5000个高品质化合物库存
应用领域
TCS JNK 5a 是一种有效的 JNK3 抑制剂,pIC50 为 6.7。TCS JNK 5a 也抑制 JNK2,pIC50为 6.5。
Cas No.: 312917-14-9
名称: N-(3-Cyano-4,5,6,7-tetrahydrobenzo[b]thienyl-2-yl)-1-naphthalenecarboxamide
别名: JNK Inhibitor IX,TCSJNK-5a)
SMILES: C1CCC2=C(C1)C(=C(S2)NC(=O)C3=CC=CC4=CC=CC=C43)C#N
分子式: C20H16N2Os
分子量: 332.4
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: JNK Inhibitor IX (TCS-JNK-5a) is a thienylnaphthamide compound that targets the ATP binding site of JNK2 and JNK3, disrupting activity with pIC50 values of 6.5 and 6.7, respectively.It demonstrates little activity against JNK1, p38α, and a panel of more than 30 other kinases (pIC50 < 5.0). For the detailed information of TCS JNK 5a(JNK Inhibitor IX), the solubility of TCS JNK 5a(JNK Inhibitor IX) in water, the solubility of TCS JNK 5a(JNK Inhibitor IX) in DMSO, the solubility of TCS JNK 5a(JNK Inhibitor IX) in PBS buffer, the animal experiment (test) of TCS JNK 5a(JNK Inhibitor IX), the cell expriment (test) of TCS JNK 5a(JNK Inhibitor IX), the in vivo, in vitro and clinical trial test of TCS JNK 5a(JNK Inhibitor IX), the EC50, IC50,and affinity,of TCS JNK 5a(JNK Inhibitor IX), For the detailed information of TCS JNK 5a(JNK Inhibitor IX), the solubility of TCS JNK 5a(JNK Inhibitor IX) in water, the solubility of TCS JNK 5a(JNK Inhibitor IX) in DMSO, the solubility of TCS JNK 5a(JNK Inhibitor IX) in PBS buffer, the animal experiment (test) of TCS JNK 5a(JNK Inhibitor IX), the cell expriment (test) of TCS JNK 5a(JNK Inhibitor IX), the in vivo, in vitro and clinical trial test of TCS JNK 5a(JNK Inhibitor IX), the EC50, IC50,and affinity,of TCS JNK 5a(JNK Inhibitor IX), Please contact DC Chemicals.
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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