首页 > 产品 > 特色产品

TCS JNK 5a(JNK Inhibitor IX)

产品编号: DC8093 Featured
TCS JNK 5a(JNK Inhibitor IX)
结构式
312917-14-9
此产品仅供科研所需，我们不出售给病人
​我们将匹配市场上最好的价格给您
Email：order@dcbio.cn
免费咨询电话：4008862077
询盘
我们的合作伙伴:
  • 20
  • 19
  • 18
  • 17
  • 16
  • 15
  • 14
  • 12
  • 11
  • 10
  • 9
  • 8
  • 13
  • 6
  • 5
  • 4
  • 3
  • 2
  • 1
中国地区超过5000个高品质化合物库存
应用领域
TCS JNK 5a 是一种有效的 JNK3 抑制剂，pIC50 为 6.7。TCS JNK 5a 也抑制 JNK2，pIC50为 6.5。
化学性质生物活性化合物的使用COA & MSDS相关产品产品说明书
Cas No.: 312917-14-9
名称: N-(3-Cyano-4,5,6,7-tetrahydrobenzo[b]thienyl-2-yl)-1-naphthalenecarboxamide
别名: JNK Inhibitor IX,TCSJNK-5a)
SMILES: C1CCC2=C(C1)C(=C(S2)NC(=O)C3=CC=CC4=CC=CC=C43)C#N
分子式: C20H16N2Os
分子量: 332.4
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: JNK Inhibitor IX (TCS-JNK-5a) is a thienylnaphthamide compound that targets the ATP binding site of JNK2 and JNK3, disrupting activity with pIC50 values of 6.5 and 6.7, respectively.It demonstrates little activity against JNK1, p38α, and a panel of more than 30 other kinases (pIC50 < 5.0). For the detailed information of TCS JNK 5a(JNK Inhibitor IX), the solubility of TCS JNK 5a(JNK Inhibitor IX) in water, the solubility of TCS JNK 5a(JNK Inhibitor IX) in DMSO, the solubility of TCS JNK 5a(JNK Inhibitor IX) in PBS buffer, the animal experiment (test) of TCS JNK 5a(JNK Inhibitor IX), the cell expriment (test) of TCS JNK 5a(JNK Inhibitor IX), the in vivo, in vitro and clinical trial test of TCS JNK 5a(JNK Inhibitor IX), the EC50, IC50,and affinity,of TCS JNK 5a(JNK Inhibitor IX), For the detailed information of TCS JNK 5a(JNK Inhibitor IX), the solubility of TCS JNK 5a(JNK Inhibitor IX) in water, the solubility of TCS JNK 5a(JNK Inhibitor IX) in DMSO, the solubility of TCS JNK 5a(JNK Inhibitor IX) in PBS buffer, the animal experiment (test) of TCS JNK 5a(JNK Inhibitor IX), the cell expriment (test) of TCS JNK 5a(JNK Inhibitor IX), the in vivo, in vitro and clinical trial test of TCS JNK 5a(JNK Inhibitor IX), the EC50, IC50,and affinity,of TCS JNK 5a(JNK Inhibitor IX), Please contact DC Chemicals.
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
产品编号 产品名称 应用领域
DC12654 PLX8394 PLX8394 是一种有效的，选择性的 BRaf 抑制剂，抑制 BRAFV600E 活性的 IC50 值约为 5 nM。
DC9743 CB1954(Tretazicar) CB1954(Tretazicar) in stock,price: 350 USD/100mg. CB1954(Tretazicar) is a anticancer prodrug that is converted in the presence of the enzyme NQO2 and co-substrate caricotamide ( EP-0152R) (EP) into a potent cytotoxic bifunctional alkylating agent.It can
DC26175 NLX-101（F-15599） NLX-101（F-15599） is a novel compound that activates serotonin 5-HT1A receptors with exceptional selectivity, having over 1000-fold higher affinity for this target over other receptors.
DC26173 YM-53601 YM-53601 is a squalene synthase inhibitor (IC50s = 79 and 90 nM in HepG2 cells and rat liver microsomes, respectively).
DC26160 Ethosalamide Etosalamide, also known as Ethosalamide, is an antipyretic and analgesics agent.
DC26155 Sulfaphenazole Sulfaphenazole is an inhibitor of CYP2C9 (Ki = 0.3 μM) that demonstrates at least 100-fold selectivity over other CYP450 isoforms (Kis = 63 and 29 μM for CYP2C8 and CYP2C18, respectively, and no activity at CYP1A1, CYP1A2, CYP3A4, CYP2C19).
DC26151 Naloxone (hydrochloride) Naloxone is an opioid inverse agonist drug used to counter the effects of opiate overdose.
DC26139 2-(5-Chloro-1H-indol-2-yl)acetic acid 2-(5-Chloro-1H-indol-2-yl)acetic acid|CAS 720000-48-6
DC12542 GOT1 inhibitor 2c GOT1抑制剂2c是谷氨酸草酰乙酸转氨酶1（GOT1）的一流的非共价抑制剂，IC50为8.2μM。
DC12541 iGOT1-01 iGOT1-01 is a small molecule inhibitor of aspartate aminotransferase 1 (glutamate oxaloacetate transaminase 1 (GOT1)) with IC50 of 11.3 uM.
​ 免费咨询电话：4008862077
​ QQ：1026657369
​ 邮箱：order@dcbio.cn
我们所有的产品仅供研究所需，严禁用于人体和其他目的
站点地图|隐私政策Copyright © 2018-2020 All Rights Reserved. 技术支持:库价软件