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TCS 5861528

产品编号: DC8262 Featured
TCS 5861528
结构式
332117-28-9
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中国地区超过5000个高品质化合物库存
应用领域
Chembridge-5861528是TRPA1离子通道阻断剂。
化学性质生物活性化合物的使用COA & MSDS相关产品产品说明书
Cas No.: 332117-28-9
名称: 2-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)-N-[4-(1-methylpropyl)phenyl]acetamide
别名: TCS 5861528,TCS-5861528,TCS5861528
SMILES: CCC(C)C1=CC=C(C=C1)NC(=O)CN2C=NC3=C2C(=O)N(C(=O)N3C)C
分子式: C19H23N5O3
分子量: 369.42
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: Selective TRPA1 channel blocker (IC50 values are 14.3 and 18.7 µM for AITC- and 4-HNE- evoked Ca2+ influx respectively). Exhibits little of no activity at TRPV1 channels. Reduces mechanical hypersensitivity, attenuates diabetes mellitus hypersensitivity and displays antinociceptive properties. For the detailed information of TCS 5861528, the solubility of TCS 5861528 in water, the solubility of TCS 5861528 in DMSO, the solubility of TCS 5861528 in PBS buffer, the animal experiment (test) of TCS 5861528, the cell expriment (test) of TCS 5861528, the in vivo, in vitro and clinical trial test of TCS 5861528, the EC50, IC50,and affinity,of TCS 5861528, For the detailed information of TCS 5861528, the solubility of TCS 5861528 in water, the solubility of TCS 5861528 in DMSO, the solubility of TCS 5861528 in PBS buffer, the animal experiment (test) of TCS 5861528, the cell expriment (test) of TCS 5861528, the in vivo, in vitro and clinical trial test of TCS 5861528, the EC50, IC50,and affinity,of TCS 5861528, Please contact DC Chemicals.
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
TITLE DOWNLOAD
MSDS_2226_DC8262_332117-28-9
COA
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