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产品编号 产品名称 CAS No.
DC4187 Docetaxel

Docetaxel, an analog of taxol, is an inhibitor of depolymerisation of microtubules through binding to stabilized microtubules.

114977-28-5
DC5099 Felbamate

Felbamate (Felbatol) is an anticonvulsant drug used in the treatment of epilepsy.

25451-15-4
DC5188 Sarecycline(P005672)

P005672 is a phase II drug for antibacterial/anti-inflammatory acne treatment.

1035979-44-2
DC5908 Honokiol

Honokiol(NSC-293100), a hydroxylated biphenyl compound isolated from the Chinese herb Magnolia officinalis, has been reported to have anticancer activities in a variety of cancer cell lines.

35354-74-6
DC6502 cardamonin

Cardamonin, isolated from the fruits of Alpinia species, is a chalconoid with anti-inflammatory and anti-tumor activity.

19309-14-9
DC6905 Linezolid (PNU-100766)

Linezolid (Zyvox) is a synthetic antibiotic used for the treatment of serious infections.

165800-03-3
DC7035 Merestinib(LY2801653 dihydrochloride)

LY2801653 2HCl is a potent, orally bioavailable, small-molecule inhibitor of c-MET kinase(Ki= 2 nM).

1206801-37-7
DC7173 Irbesartan

Irbesartan is a highly potent and specific angiotensin II type 1 (AT1) receptor antagonist with IC50 of 1.3 nM.

138402-11-6
DC7204 Ezatiostat(TER199; TLK199)

Ezatiostat(TER199; TLK199) is a glutathione analog inhibitor of glutathione S-transferase (GST) P1-1.

168682-53-9
DC7222 P005091(P5091)

P005091(P5091) is a selective and potent inhibitor of ubiquitin-specific protease 7 (USP7) with EC50 of 4.2 μM.

882257-11-6
DC7301 SSR128129E

SSR128129E is an orally-active and allosteric FGFR1 inhibitor with IC50 of 1.9 μM, while not affecting other related RTKs.

848318-25-2
DC7323 Pritelivir(BAY-57-1293)

BAY 57-1293 represents a new class of potent inhibitors of herpes simplex virus (HSV) that target the virus helicase primase complex.

348086-71-5
DC7368 AZD5363

AZD5363, a novel pyrrolopyrimidine-derived compound, inhibits all AKT isoforms (IC50 <10 nM).

1143532-39-1
DC7455 Lonafarnib

Lonafarnib(Sch66336) is an orally bioavailable FPTase inhibitor for H-ras, K-ras-4B and N-ras with IC50 of 1.9 nM, 5.2 nM and 2.8 nM, respectively.

193275-84-2
DC7500 Siramesine-hydrochloride

Siramesine(Lu 28-179) Hcl is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of cancer cells and to exhibit a potent anticancer activity in vivo.

224177-60-0
DC7546 LHW090-A7

For the detailed information of LHW090-A7, the solubility of LHW090-A7 in water, the solubility of LHW090-A7 in DMSO, the solubility of LHW090-A7 in PBS buffer, the animal experiment (test) of LHW090-A7, the cell expriment (test) of LHW090-A7, the in viv

1308256-94-1
DC7551 RG3039(PF-06687859)

For the detailed information of PF-0668759, the solubility of PF-0668759 in water, the solubility of PF-0668759 in DMSO, the solubility of PF-0668759 in PBS buffer, the animal experiment (test) of PF-0668759, the cell expriment (test) of PF-0668759, the

1005504-62-0
DC7619 Tazarotenic acid (AGN 190299)

Tazarotenic Acid is an agent that acts as the principle active metabolite

118292-41-4
DC7635 IB-MECA

IB-MECA is a potent and selective A3 adenosine receptor agonist (Ki values are 1.1, 54 and 56 nM for A3, A1 and A2A receptors respectively).

152918-18-8
DC7708 UNBS5162

UNBS5162 is a novel naphthalimide that decreases CXCL chemokine expression in experimental prostate cancers; the mean antiproliferative activity IC50 value is 17.9 uM for 9 cancer cell lines; hydrolysis product of UNBS3157.

956590-23-1
DC7727 PH-797804

PH-797804 is a potent and selective p38 inhibitor with IC50 of 26 nM.

586379-66-0
DC7745 Filorexant(mk-6096)

MK-6096 is an orally bioavailable potent and selective reversible antagonist of OX(1)R and OX(2)R currently in clinical development for insomnia.

1088991-73-4
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