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产品编号 产品名称 CAS No.
DC10622 S38093

S 38093 是一种大脑渗透的 H3 receptor 拮抗剂,对大鼠,小鼠和人的 H3 受体具有不同的亲和力,Ki 值分别为 8.8,1.44 和 1.2 µM。

862896-30-8
DC10623 AG-494

2-cyano-3-(3,4-dihydroxyphenyl)-N-phenylprop-2-enamide

133550-35-3
DC10624 Targocil

Targocil 可用作磷壁酸 (WTA) 生物合成的抑菌抑制剂,可抑制甲氧西林敏感金黄色葡萄球菌 (MSSA)和耐甲氧西林金黄色葡萄球菌 (MRSA) 的生长,对于 MRSA 和 MSSA 的 MIC90 值都为 2 μg/mL。

1200443-21-5
DC10638 ZK756326 2HCl

2-[2-[4-[(3-苯氧基苯基)甲基]-1-哌嗪基]乙氧基]乙醇

874911-96-3
DC1064 RITA (NSC652287)

RITA 是一种有效的 p53-HDM-2 相互作用抑制剂,可与 p53dN 结合,Kd 值为 1.5 nM,同时能够诱导 DNA-DNA 交联。

213261-59-7
DC10650 MDVN1003

MDVN1003是BTK和PI3Kδ的有效抑制剂。

2058116-52-0
DC10652 HG-14-10-04

HG-14-10-04是特异的ALK抑制剂,IC50为20 nM。

1356962-34-9
DC10653 TLR7-IN-1

TLR7 agonist 2 是一种有效且有选择性的 Toll 样受体 7 (TLR7) 激动剂,LEC 值为 0.4 μM。

1642857-69-9
DC10655 BETA-GUANIDINOPROPIONIC ACID

BETA-GUANIDINOPROPIONIC ACID用作食品、饮料、饲料添加剂,营养强化剂,化妆品用表面活性剂和医药原料等

353-09-3
DC10667 Gea3162

3-(3,4-dichlorophenyl)-1-oxa-2-aza-3-azonia-4-azanidacyclopent-2-en-5-imine

144576-10-3
DC10668 GYY4137 morpholine salt

(4-甲氧基苯基)吗啉基-二硫代膦酸与吗啉的化合物,

106740-09-4
DC10669 KYP-2047

KYP-2047 is a very potent, selective inhibitor of Prolyl oligopeptidase (POP), also known as prolyl endopeptidase (PEP or PE). Ki = .023nM (porcine).

796874-99-2
DC10674 1-EBIO

1-EBIO is an Epithelial KCa channel activator. Promotes ESC differentiation into cardiomyocytes.

10045-45-1
DC10676 Z-IETD-pNA(GRANZYME B SUBSTRATE I)

Z-IETD-pNA is a colorimetric caspase-8/granzyme B substrate containing the benzyloxycarbonyl (Z) moiety.

498555-58-1
DC10678 Fluticasone

Fluticasone是糖皮质激素受体(GR)激动剂。

90566-53-3
DC10682 Velaresol

5-(2-Formyl-3-hydroxyphenoxy)pentanoic acid

77858-21-0
DC10684 QCC-374

7,8-二氢-2,3-二(4-甲基苯基)吡啶并[2,3-b]吡嗪-5(6H)-庚酸

1356331-63-9
DC10685 Adipamidoxime(NSC 70868)

Adipamidoxime(NSC 70868) is a new bioactive compoud.

15347-78-1
DC10686 Cosan-528

N-(4-溴-2-甲基苯基)-2-氯乙酰胺,

96686-51-0
DC10687 Sematilide hydrochloride

Sematilide, also known as CK-1752, is a class III antiarrhythmic.

101526-62-9
DC10690 SPI-112Me

SPI-112Me is a prodrug for SPI-112, which preferentially inhibits the PTPase activity of Shp2 over Shp1 and PTP1B by a factor of 20 in cell-free assays.

1243685-62-2
DC10691 Pyronaridine

4-[(7-chloro-2-methoxy-1,5-dihydrobenzo[b][1,5]naphthyridin-10-yl)imino]-2,6-bis(pyrrolidin-1-ylmethyl)cyclohexa-2,5-dien-1-one

74847-35-1
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