Gilteritinib(ASP2215)

产品编号: DC8164 Featured
Gilteritinib(ASP2215)
结构式
1254053-43-4
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中国地区超过5000个高品质化合物库存
应用领域
Gilteritinib 是一种有效的 FLT3/AXL 抑制剂,IC50 分别为 0.29 nM/0.73 nM。
Cas No.: 1254053-43-4
名称: 6-ethyl-3-({3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}amino)-5-[(tetrahydro-2H-pyran-4-yl)amino]pyrazine-2-carboxamide
别名: ASP2215
SMILES: NC(C1=NC(CC)=C(NC2CCOCC2)N=C1NC3=CC(OC)=C(N4CCC(N5CCN(C)CC5)CC4)C=C3)=O
分子式: C29H44N8O3
分子量: 552.35
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: For the detailed information of Gilteritinib(ASP2215), the solubility of Gilteritinib(ASP2215) in water, the solubility of Gilteritinib(ASP2215) in DMSO, the solubility of Gilteritinib(ASP2215) in PBS buffer, the animal experiment (test) of Gilteritinib(ASP2215), the cell expriment (test) of Gilteritinib(ASP2215), the in vivo, in vitro and clinical trial test of Gilteritinib(ASP2215), the EC50, IC50,and affinity,of Gilteritinib(ASP2215), For the detailed information of Gilteritinib(ASP2215), the solubility of Gilteritinib(ASP2215) in water, the solubility of Gilteritinib(ASP2215) in DMSO, the solubility of Gilteritinib(ASP2215) in PBS buffer, the animal experiment (test) of Gilteritinib(ASP2215), the cell expriment (test) of Gilteritinib(ASP2215), the in vivo, in vitro and clinical trial test of Gilteritinib(ASP2215), the EC50, IC50,and affinity,of Gilteritinib(ASP2215), Please contact DC Chemicals.
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
产品编号 产品名称 应用领域
DC8164 Gilteritinib(ASP2215) Gilteritinib 是一种有效的 FLT3/AXL 抑制剂,IC50 分别为 0.29 nM/0.73 nM。
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