Bazedoxifene-Acetate
产品编号: DC7372
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应用领域
Bazedoxifene acetate (TSE-424 acetate) 是第三代选择性雌激素受体调节剂 (SERM)， IC50分别为26和99 nM。
| Cas No.: |
198481-33-3 |
| 名称: |
acetic acid;1-[[4-[2-(azepan-1-yl)ethoxy]phenyl]methyl]-2-(4-hydroxyphenyl)-3-methylindol-5-ol |
| 别名: |
TSE 424; Viviant; WAY-TES 424 |
| SMILES: |
CC1=C(N(C2=C1C=C(C=C2)O)CC3=CC=C(C=C3)OCCN4CCCCCC4)C5=CC=C(C=C5)O.CC(=O)O |
| 分子式: |
C32H38N2O5 |
| 分子量: |
530.65452 |
| 纯度: |
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| 保存条件: |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: |
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| In Vitro: |
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| References: |
Bazedoxifene is a third generation selective estrogen receptor modulator (SERM). Bazedoxifene does not stimulate ERα mediated transcriptional activity and acts as an antagonist to estradiol in cultured breast cancer (bMCF-7) cells. Similar results are see |
| Kinase Assay: |
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| Cell Assay: |
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| Animal Administration: |
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| References: |
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MSDS
COA
| LOT NO. |
DOWNLOAD |
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| 2018-0101 |
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询盘
