Lasmiditan (COL-144; LY573144)
产品编号: DC7710
我们的合作伙伴:
中国地区超过5000个高品质化合物库存
应用领域
Lasmiditan (COL-144; LY573144) is a high-affinity, highly selective 5-HT1F receptor agonist(Ki=2.1 nM), compared with Ki of 1043 nM and 1357 nM at the 5-HT(1B) and 5-HT(1D) receptors, respectively.
| Cas No.: |
439239-90-4 |
| 名称: |
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| 别名: |
COL-144; LY-573144,COL144; LY 573144 |
| SMILES: |
FC1=CC(F)=C(C(NC2=CC=CC(C(C3CCN(C)CC3)=O)=N2)=O)C(F)=C1 |
| 分子式: |
C19H18F3N3O2 |
| 分子量: |
377.36 |
| 纯度: |
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| 保存条件: |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: |
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| References: |
Lasmiditan (COL-144; LY573144) is a high-affinity, highly selective 5-HT1F receptor agonist(Ki=2.1 nM), compared with Ki of 1043 nM and 1357 nM at the 5-HT(1B) and 5-HT(1D) receptors, respectively.
IC50 value: 2.1 nM (Ki, 5-HT1F); >1000 nM (Ki, 5-HT1B/5- |
| Kinase Assay: |
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| Animal Administration: |
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| References: |
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MSDS
| TITLE |
DOWNLOAD |
| MSDS_3451_DC7710_439239-90-4 |
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COA
| LOT NO. |
DOWNLOAD |
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