ACT058362 (Palosuran)
产品编号: DC7970
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应用领域
Palosuran (ACT-058362)是高活性人UT受体特异性拮抗剂，IC50为3.6 nM。
| Cas No.: |
540769-28-6 |
| 名称: |
Urea, N-[2-[4-hydroxy-4-(phenylMethyl)-1-piperidinyl]ethyl]-N'-(2-Methyl-4-quinolinyl)- |
| 别名: |
ACT058362，ACT-058362 |
| SMILES: |
N(CCN1CCC(O)(CC2=CC=CC=C2)CC1)C(NC1C2C(N=C(C)C=1)=CC=CC=2)=O |
| 分子式: |
C25H30N4O2 |
| 分子量: |
418.53 |
| 纯度: |
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| 保存条件: |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: |
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| In Vitro: |
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| References: |
Palosuran inhibited 125I-U-II binding to human UT receptors in membrane preparations from CHO cells carrying the human UT receptors almost as potently as cold U-II, with an IC50 of 3.6 ± 0.2 nM. On cells, the inhibitory binding potency of palosuran agains |
| Kinase Assay: |
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| Cell Assay: |
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| Animal Administration: |
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| References: |
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MSDS
| TITLE |
DOWNLOAD |
| MSDS_2048_DC7970_540769-28-6 |
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COA
| LOT NO. |
DOWNLOAD |
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