Otenabant (CP-945598 free base)
产品编号: DC7109
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应用领域
Otenabant 是一种有效的，选择性的 cannabinoid receptor CB1 拮抗剂，Ki 值为 0.7 nM，对其选择性是对 CB2 的 1000 多倍。
| Cas No.: |
686344-29-6 |
| 名称: |
1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)purin-6-yl]-4-(ethylamino)piperidine-4-carboxamide |
| 别名: |
CP 945598; CP-945598; CP945598 |
| SMILES: |
N(C1=C2C(=NC=N1)N(C1=CC=C(Cl)C=C1)C(C1=CC=CC=C1Cl)=N2)1CCC(NCC)(C(N)=O)CC1 |
| 分子式: |
C25H25Cl2N7O |
| 分子量: |
510.41 |
| 纯度: |
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| 保存条件: |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: |
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| References: |
CP-945598 inhibits CB1 receptor with moderate unbound microsomal clearance, low hERG Affinity and adequate CNS penetration. CP-945598 has low affinity with Ki of 7.6 μM For human CB2 receptors. CP-945598 reverses four cannabinoid agonistmediated behavio |
| Kinase Assay: |
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| Animal Administration: |
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| References: |
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MSDS
COA
| LOT NO. |
DOWNLOAD |
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| 2018-0101 |
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询盘
