Almorexant HCl (Act-078573)
产品编号: DC7692
Featured
我们的合作伙伴:
中国地区超过5000个高品质化合物库存
应用领域
Almorexant hydrochloride (ACT 078573 hydrochloride) 是一种有效的食欲素受体 orexin 1 receptor (OX1)/orexin 2 receptor (OX2) 拮抗剂,Ki 分别为 1.3 和 0.17 nM。
| Cas No.: |
913358-93-7 |
| 名称: |
|
| 别名: |
ACT-078573; ACT 078573; ACT078573 |
| SMILES: |
C(NC)(=O)[C@@H](N1CCC2=C([C@H]1CCC1=CC=C(C(F)(F)F)C=C1)C=C(OC)C(OC)=C2)C1=CC=CC=C1.[H]Cl |
| 分子式: |
C29H32ClF3N2O3 |
| 分子量: |
549.02 |
| 纯度: |
|
| 保存条件: |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: |
|
| In Vivo: |
|
| In Vitro: |
|
| References: |
Almorexant(ACT078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.
IC50 value: 1.3/0.7 nM(OX1/OX2 receptor)
Target: Dual OX!/OX2 receptor
in |
| Kinase Assay: |
|
| Cell Assay: |
|
| Animal Administration: |
|
| References: |
|
MSDS
| TITLE |
DOWNLOAD |
| MSDS_1906_DC7692_913358-93-7 |
|
COA
| LOT NO. |
DOWNLOAD |
|
|
询盘