Endoxifen

产品编号: DC8265 Featured
Endoxifen
结构式
110025-28-0
此产品仅供科研所需,我们不出售给病人
​我们将匹配市场上最好的价格给您
Email:order@dcbio.cn
免费咨询电话:4008862077
我们的合作伙伴:
  • 20
  • 19
  • 18
  • 17
  • 16
  • 15
  • 14
  • 12
  • 11
  • 10
  • 9
  • 8
  • 13
  • 6
  • 5
  • 4
  • 3
  • 2
  • 1
中国地区超过5000个高品质化合物库存
应用领域
Endoxifen 是tamoxifen 的关键活性代谢物,与雌激素受体 (estrogen receptor) 有较高的亲和力和特异性,同时也能抑制芳香酶的活性。
Cas No.: 110025-28-0
名称: (E/Z)-4-[1-[4-[2-(Methylamino)ethoxy]phenyl]-2-phenyl-1-buten-1-yl]-phenol
别名:
SMILES: CC/C(=C(/C1=CC=C(C=C1)O)\C2=CC=C(C=C2)OCCNC)/C3=CC=CC=C3
分子式: C25H27NO2
分子量: 373.49
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: Endoxifen is a Estrogen receptor α (ERα) ligand; potent antiestrogen,an active metabolite of the cancer drug tamoxifen.Primary metabolite responsible for the effectiveness of tamoxifen in ER-positive breast cancer. For the detailed information of Endoxifen, the solubility of Endoxifen in water, the solubility of Endoxifen in DMSO, the solubility of Endoxifen in PBS buffer, the animal experiment (test) of Endoxifen, the cell expriment (test) of Endoxifen, the in vivo, in vitro and clinical trial test of Endoxifen, the EC50, IC50,and affinity,of Endoxifen, For the detailed information of Endoxifen, the solubility of Endoxifen in water, the solubility of Endoxifen in DMSO, the solubility of Endoxifen in PBS buffer, the animal experiment (test) of Endoxifen, the cell expriment (test) of Endoxifen, the in vivo, in vitro and clinical trial test of Endoxifen, the EC50, IC50,and affinity,of Endoxifen, Please contact DC Chemicals.
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
产品编号 产品名称 应用领域
DC9268 AZD9496 AZD9496 是有效,选择性的雌激素受体 (ERα) 拮抗剂,IC50 为 0.28 nM。AZD9496 是一种口服有效的选择性雌激素受体降解剂 (SERD)
DC8265 Endoxifen Endoxifen 是tamoxifen 的关键活性代谢物,与雌激素受体 (estrogen receptor) 有较高的亲和力和特异性,同时也能抑制芳香酶的活性。
DC8049 SNG-1153 SNG1153是一种合成的ER - α36调节剂,在体内外都具有作用活性。
DC10832 (E/Z)-4-hydroxy Tamoxifen (E/Z)-4-Hydroxytamoxifen 是 (Z)-4-Hydroxytamoxifen 和 (E)-4-Hydroxytamoxifen 的消旋体。(E/Z)-4-Hydroxytamoxifen 是雌激素受体 (estrogen receptor) 调节剂。
DC10755 LSZ102 LSZ-102 是一种强效, 口服生物有效的选择性雌激素受体降解剂, 其 IC50 值为 0.2 nM。