PX 12

产品编号: DC7992 Featured
PX 12
结构式
141400-58-0
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中国地区超过5000个高品质化合物库存
应用领域
PX-12(IV-2) is an irreversible inhibitor of Thioredoxin-1(Trx-1) currently in clinical development as an antitumor agent; IC50=7 uM in Hela, MTT assay, 72 h.
Cas No.: 141400-58-0
名称: 2-[(1-Methylpropyl)dithio]-1H-imidazole; IV-2
别名: PX-12,PX12
SMILES: CCC(SSC1=NC=CN1)C
分子式: C7H12N2S2
分子量: 188.31
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: PX-12(IV-2) is an irreversible inhibitor of Thioredoxin-1(Trx-1) currently in clinical development as an antitumor agent; IC50=7 uM in Hela, MTT assay, 72 h.Based on MTT assays, PX-12 inhibited the growth of HeLa cells with an IC50 value of ~7 μM at 72 h.
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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