| Cas No.: | 372196-77-5 |
| 名称: | (E)-N'-((6-bromoH-imidazo[1,2-a]pyridin-3-yl)methylene)-N,2-dimethyl-5-nitrobenzenesulfonohydrazidehydrochloride |
| 别名: | PIK-75 Hydrochloride; PIK 75 |
| SMILES: | CC1=C(C=C(C=C1)[N+](=O)[O-])S(=O)(=O)N(C)/N=C/C2=CN=C3N2C=C(C=C3)Br.Cl |
| 分子式: | C16H14BrN5O4S |
| 分子量: | 452.282 |
| 纯度: | |
| 保存条件: | 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: | |
| In Vivo: | |
| In Vitro: | |
| References: | PIK-75 shows the impressive potency and iso Form selectivity at p110α while the corresponding IC50 values are 1300 nM, 76 nM and 510 nM For other PI3K iso Forms, p110β, -γ, and -δ, respectively. Furthermore, when binding to purified p110α, PIK-75 is a no |
| Kinase Assay: | |
| Cell Assay: | |
| Animal Administration: | |
| References: |
MSDS
COA
| LOT NO. | DOWNLOAD |
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| 2018-0101 |
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