| Cas No.: | 702675-74-9 |
| 名称: | N-(3-(5-iodo-4-(3-(thiophene-2-carboxamido)propylamino)pyrimidin-2-ylamino)phenyl)pyrrolidine-1-carboxamide |
| 别名: | BX 795; BX-795 |
| SMILES: | N(C(NC1=CC=CC(NC2=NC=C(I)C(NCCCNC(C3SC=CC=3)=O)=N2)=C1)=O)1CCCC1 |
| 分子式: | C23H26In7O2S |
| 分子量: | 591.47 |
| 纯度: | |
| 保存条件: | 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: | |
| In Vivo: | |
| In Vitro: | |
| References: | BX-795 effectively blocks PDK1 activity in PC-3 cells, as shown by their ability to block phosphorylation of S6K1, Akt, PKCδ, and GSK3β. BX-795 potently inhibits tumor cell growth on plastic with IC50 of 1.6, 1.4, and 1.9 μM For MDA-468, HCT-116 and MiaP |
| Kinase Assay: | |
| Cell Assay: | |
| Animal Administration: | |
| References: |
MSDS
COA
| LOT NO. | DOWNLOAD |
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| 2018-0101 |
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